FI (list display)

  • A61K31/00
  • Medicinal preparations containing organic active ingredients [2] HB CC 4C206
  • A61K31/01
  • .Hydrocarbons [2] HB CC 4C206
  • A61K31/015
  • ..carbocyclic [2] HB CC 4C206
  • A61K31/02
  • .Halogenated hydrocarbons [2] HB CC 4C206
  • A61K31/025
  • ..carbocyclic [2] HB CC 4C206
  • A61K31/03
  • ...aromatic [2] HB CC 4C206
  • A61K31/035
  • ..having aliphatic unsaturation [2] HB CC 4C206
  • A61K31/04
  • .Nitro compounds [2] HB CC 4C206
  • A61K31/045
  • .Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates (hydroperoxides A61K 31/327) [2,7] HB CC 4C206
  • A61K31/047
  • ..having two or more hydroxy groups, e.g. sorbitol [7] HB CC 4C206
  • A61K31/05
  • ..Phenols [2] HB CC 4C206
  • A61K31/055
  • ...the aromatic ring being substituted by halogen [2] HB CC 4C206
  • A61K31/06
  • ...the aromatic ring being substituted by nitro groups [2] HB CC 4C206
  • A61K31/065
  • ..Diphenyl-substituted acyclic alcohols [2] HB CC 4C206
  • A61K31/07
  • ..Retinol compounds, e.g. vitamin A (retinoic acids A61K 31/203) [2,7] HB CC 4C206
  • A61K31/075
  • .Ethers or acetals [2] HB CC 4C206
  • A61K31/08
  • ..acyclic, e.g. paraformaldehyde [2] HB CC 4C206
  • A61K31/085
  • ..having an ether linkage to aromatic ring nuclear carbon [2] HB CC 4C206
  • A61K31/09
  • ...having two or more such linkages [2] HB CC 4C206
  • A61K31/095
  • .Sulfur, selenium or tellurium compounds, e.g. thiols [2] HB CC 4C206
  • A61K31/10
  • ..Sulfides; Sulfoxides; Sulfones [2] HB CC 4C206
  • A61K31/105
  • ..Persulfides (thiuram disulfides A61K 31/145; thiosulfonic acids A61K 31/185) [2] HB CC 4C206
  • A61K31/11
  • .Aldehydes [2] HB CC 4C206
  • A61K31/115
  • ..Formaldehyde [2] HB CC 4C206
  • A61K31/12
  • .Ketones [2] HB CC 4C206
  • A61K31/121
  • ..acyclic [7] HB CC 4C206
  • A61K31/122
  • ..having the oxygen atom directly attached to a ring, e.g. quinones, vitamin K1, anthralin [7] HB CC 4C206
  • A61K31/125
  • ...Camphor; Nuclear substituted derivatives thereof [2] HB CC 4C206
  • A61K31/13
  • .Amines, e.g. amantadine (A61K 31/04 takes precedence) [2] HB CC 4C206
  • A61K31/131
  • ..acyclic [7] HB CC 4C206
  • A61K31/132
  • ..having two or more amino groups, e.g. spermidine, putrescine [7] HB CC 4C206
  • A61K31/133
  • ..having hydroxy groups, e.g. sphingosine [7] HB CC 4C206
  • A61K31/135
  • ..having aromatic rings, e.g. methadone [2,7] HB CC 4C206
  • A61K31/136
  • ...having the amino group directly attached to the aromatic ring, e.g. benzeneamine [7] HB CC 4C206
  • A61K31/137
  • ...Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine [7] HB CC 4C206
  • A61K31/138
  • ...Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine (atenolol A61K 31/165; pindolol A61K 31/404; timolol A61K 31/5377) [7] HB CC 4C206
  • A61K31/14
  • ..Quaternary ammonium compounds, e.g. edrophonium, choline (betaines A61K 31/205) [2] HB CC 4C206
  • A61K31/145
  • ..having sulfur atoms, e.g. thiurams (2) (isothioureas A61K 31/155) [2,7] HB CC 4C206
  • A61K31/15
  • ..Oximes ( HB CC 4C206
  • A61K31/155
  • ..Amidines ([figure]), e.g. guanidine (H2N—C(=NH)—NH2), isourea (HN=C(OH)NH2), isothiourea (HN=C(SH)—NH2) [2] HB CC 4C206
  • A61K31/16
  • .Amides, e.g. hydroxamic acids [2] HB CC 4C206
  • A61K31/164
  • ..of a carboxylic acid with an aminoalcohol, e.g. ceramides [7] HB CC 4C206
  • A61K31/165
  • ..having aromatic rings, e.g. colchicine, atenolol, progabide [2] HB CC 4C206
  • A61K31/166
  • ...having the carbon atom of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol [7] HB CC 4C206
  • A61K31/167
  • ...having the nitrogen atom of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol [7] HB CC 4C206
  • A61K31/17
  • ..having the group HB CC 4C206
  • A61K31/175
  • ...having the group [figure], figure], e.g. carbonohydrazides, carbazones, semicarbazides, semicarbazones; Thioanalogues thereof [2,7] HB CC 4C206
  • A61K31/18
  • ..Sulfonamides (compounds containing a para-N-benzene-sulfonyl-N-group A61K 31/63) [2] HB CC 4C206
  • A61K31/185
  • .Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids (hydroxamic acids A61K 31/16; peroxy acids A61K 31/327) [2,7] HB CC 4C206
  • A61K31/19
  • ..Carboxylic acids, e.g. valproic acid (salicylic acid A61K 31/60) [2,7] HB CC 4C206
  • A61K31/191
  • ...Acyclic acids having two or more hydroxy groups, e.g. gluconic acid [7] HB CC 4C206
  • A61K31/192
  • ...having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid [7] HB CC 4C206
  • A61K31/194
  • ...having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid [7] HB CC 4C206
  • A61K31/195
  • ...having an amino group HB CC 4C206
  • A61K31/196
  • ....the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil [7] HB CC 4C206
  • A61K31/197
  • ....the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid (carnitine A61K 31/205) [2006.01] HB CC 4C206
  • A61K31/198
  • .....Alpha-amino acids, e.g. alanine or edetic acid [EDTA] (betaine A61K 31/205; proline A61K 31/401; tryptophan A61K 31/405; histidine A61K 31/4172; peptides not degraded to individual amino acids A61K 38/00) [2006.01] HB CC 4C206
  • A61K31/20
  • ...having a carboxyl group bound to an acyclic chain of seven or more carbon atoms, e.g. stearic, palmitic or arachidic acid [2] HB CC 4C206
  • A61K31/201
  • ....having one or two double bonds, e.g. oleic or linoleic acid [7] HB CC 4C206
  • A61K31/202
  • ....having three or more double bonds, e.g. linolenic acid (eicosanoids, e.g. leukotrienes, A61K 31/557) [7] HB CC 4C206
  • A61K31/203
  • ....Retinoic acids [7] HB CC 4C206
  • A61K31/205
  • ..Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine [2] HB CC 4C206
  • A61K31/21
  • .Esters, e.g. nitroglycerine, selenocyanates [2] HB CC 4C206
  • A61K31/215
  • ..of carboxylic acids [2] HB CC 4C206
  • A61K31/216
  • ...of acids having aromatic rings, e.g. benactizyne, clofibrate [7] HB CC 4C206
  • A61K31/22
  • ...of acyclic acids, e.g. pravastatin [2] HB CC 4C206
  • A61K31/221
  • ....with compounds having an amino group, e.g. acetylcholine, acetylcarnitine [7] HB CC 4C206
  • A61K31/222
  • ....with compounds having aromatic groups, e.g. dipivefrine, ibopamine [7] HB CC 4C206
  • A61K31/223
  • ....of alpha-amino acids [7] HB CC 4C206
  • A61K31/225
  • ....Polycarboxylic acids [2] HB CC 4C206
  • A61K31/23
  • ....of acids having a carboxyl group bound to a chain of seven or more carbon atoms [2] HB CC 4C206
  • A61K31/231
  • .....having one or two double bonds [7] HB CC 4C206
  • A61K31/232
  • .....having three or more double bonds, e.g. etretinate [7] HB CC 4C206
  • A61K31/235
  • ...having an aromatic ring attached to a carboxyl group [2] HB CC 4C206
  • A61K31/24
  • ....having an amino or nitro group [2] HB CC 4C206
  • A61K31/245
  • .....Amino benzoic acid types, e.g. procaine, novocaine (salicylic acid esters A61K 31/60) [2] HB CC 4C206
  • A61K31/25
  • ...with polyoxyalkylated alcohols, e.g. esters of polyethylene glycol [2] HB CC 4C206
  • A61K31/255
  • ..of sulfoxy acids or sulfur analogues thereof [2] HB CC 4C206
  • A61K31/26
  • ..Cyanate or isocyanate esters; Thiocyanate or isothiocyanate esters [2,7] HB CC 4C206
  • A61K31/265
  • ..of carbonic, thiocarbonic or thiocarboxylic acids, e.g. thioacetic acid, xanthogenic acid, trithiocarbonic acid [2] HB CC 4C206
  • A61K31/27
  • ..of carbamic or thiocarbamic acids, e.g. meprobamate, carbachol, neostigmine [2] HB CC 4C206
  • A61K31/275
  • .Nitriles; Isonitriles [2] HB CC 4C206
  • A61K31/277
  • ..having a ring, e.g. verapamil [7] HB CC 4C206
  • A61K31/28
  • .Compounds containing heavy metals [2] HB CC 4C206
  • A61K31/282
  • ..Platinum compounds [7] HB CC 4C206
  • A61K31/285
  • ..Arsenic compounds [2] HB CC 4C206
  • A61K31/29
  • ..Antimony or bismuth compounds [2] HB CC 4C206
  • A61K31/295
  • ..Iron group metal compounds [2] HB CC 4C206
  • A61K31/30
  • ..Copper compounds [2] HB CC 4C206
  • A61K31/305
  • ..Mercury compounds [2] HB CC 4C206
  • A61K31/31
  • ...containing nitrogen [2] HB CC 4C206
  • A61K31/315
  • ..Zinc compounds [2] HB CC 4C206
  • A61K31/32
  • ..Tin compounds [2] HB CC 4C206
  • A61K31/325
  • .Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof (thiurams A61K 31/145) [2] HB CC 4C206
  • A61K31/327
  • .Peroxy compounds, e.g. hydroperoxides, peroxides, peroxy acids [7] HB CC 4C206
  • A61K31/33
  • .Heterocyclic compounds [2] HB CC 4C086
  • A61K31/335
  • ..having oxygen as the only ring hetero atom, e.g. fungichromin [2] HB CC 4C086
  • A61K31/336
  • ...having three-membered rings, e.g. oxirane, fumagillin [7] HB CC 4C086
  • A61K31/337
  • ...having four-membered rings, e.g. taxol [7] HB CC 4C086
  • A61K31/34
  • ...having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide [2] HB CC 4C086
  • A61K31/341
  • ....not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine [7] HB CC 4C086
  • A61K31/343
  • ....condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone [7] HB CC 4C086
  • A61K31/345
  • ....Nitrofurans (nitrofurantoin A61K 31/4178) [2,7] HB CC 4C086
  • A61K31/35
  • ...having six-membered rings with one oxygen as the only ring hetero atom [2] HB CC 4C086
  • A61K31/351
  • ....not condensed with another ring [7] HB CC 4C086
  • A61K31/352
  • ....condensed with carbocyclic rings, e.g. cannabinols, methantheline [7] HB CC 4C086
  • A61K31/353
  • .....3,4-Dihydrobenzopyrans, e.g. chroman, catechin [7] HB CC 4C086
  • A61K31/355
  • ......Tocopherols, e.g. vitamin E [2] HB CC 4C086
  • A61K31/357
  • ...having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel [7] HB CC 4C086
  • A61K31/36
  • ....Compounds containing methylenedioxyphenyl groups, e.g. sesamin [2] HB CC 4C086
  • A61K31/365
  • ...Lactones [2] HB CC 4C086
  • A61K31/366
  • ....having six-membered rings, e.g. delta-lactones [7] HB CC 4C086
  • A61K31/37
  • .....Coumarins, e.g. psoralen [2] HB CC 4C086
  • A61K31/375
  • ....Ascorbic acid, i.e. vitamin C; Salts thereof [2] HB CC 4C086
  • A61K31/38
  • ..having sulfur as a ring hetero atom [2] HB CC 4C086
  • A61K31/381
  • ...having five-membered rings [7] HB CC 4C086
  • A61K31/382
  • ...having six-membered rings, e.g. thioxanthenes (thiothixene A61K 31/496) [7] HB CC 4C086
  • A61K31/385
  • ...having two or more sulfur atoms in the same ring [2] HB CC 4C086
  • A61K31/39
  • ...having oxygen atoms in the same ring [2] HB CC 4C086
  • A61K31/395
  • .. having nitrogen as a ring hetero atom e.g. guanethidine or rifamycins HB CC 4C086
  • A61K31/396
  • ...having three-membered rings, e.g. aziridine [7] HB CC 4C086
  • A61K31/397
  • ...having four-membered rings, e.g. azetidine [7] HB CC 4C086
  • A61K31/40
  • ...having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil [2] HB CC 4C086
  • A61K31/401
  • ....Proline; Derivatives thereof, e.g. captopril [7] HB CC 4C086
  • A61K31/4015
  • ....having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide [7] HB CC 4C086
  • A61K31/402
  • ....1-aryl-substituted, e.g. piretanide [7] HB CC 4C086
  • A61K31/4025
  • ....not condensed and containing further heterocyclic rings, e.g. cromakalim [7] HB CC 4C086
  • A61K31/403
  • ....condensed with carbocyclic rings, e.g. carbazole [7] HB CC 4C086
  • A61K31/4035
  • .....Isoindoles, e.g. phthalimide [7] HB CC 4C086
  • A61K31/404
  • .....Indoles, e.g. pindolol [7] HB CC 4C086
  • A61K31/4045
  • ......Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin [7] HB CC 4C086
  • A61K31/405
  • ......Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin [2] HB CC 4C086
  • A61K31/407
  • ....condensed with heterocyclic ring systems, e.g. ketorolac, physostigmine [7] HB CC 4C086
  • A61K31/409
  • ....having four such rings, e.g. porphine derivatives, bilirubin, biliverdine (hemin, hematin A61K 31/555) [7] HB CC 4C086
  • A61K31/41
  • ...having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole [2] HB CC 4C086
  • A61K31/415
  • ....1,2-Diazoles [2,7] HB CC 4C086
  • A61K31/4152
  • .....having oxo groups directly attached to the heterocyclic ring, e.g. antipyrine, phenylbutazone, sulfinpyrazone [7] HB CC 4C086
  • A61K31/4155
  • .....not condensed and containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/416
  • .....condensed with carbocyclic ring systems, e.g. indazole [7] HB CC 4C086
  • A61K31/4162
  • .....condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/4164
  • ....1,3-Diazoles [7] HB CC 4C086
  • A61K31/4166
  • .....having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin [7] HB CC 4C086
  • A61K31/4168
  • .....having a nitrogen atom attached in position 2, e.g. clonidine [7] HB CC 4C086
  • A61K31/417
  • .....Imidazole-alkylamines, e.g. histamine, phentolamine [7] HB CC 4C086
  • A61K31/4172
  • .....Imidazole-alkanecarboxylic acids, e.g. histidine [7] HB CC 4C086
  • A61K31/4174
  • .....Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole [7] HB CC 4C086
  • A61K31/4178
  • .....not condensed and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin [7] HB CC 4C086
  • A61K31/4184
  • .....condensed with carbocyclic rings, e.g. benzimidazoles [7] HB CC 4C086
  • A61K31/4188
  • .....condensed with heterocyclic ring systems, e.g. biotin, sorbinil [7] HB CC 4C086
  • A61K31/4192
  • ....1,2,3-Triazoles [7] HB CC 4C086
  • A61K31/4196
  • ....1,2,4-Triazoles [7] HB CC 4C086
  • A61K31/42
  • ....Oxazoles [2,7] HB CC 4C086
  • A61K31/421
  • .....1,3-Oxazoles, e.g. pemoline, trimethadione [7] HB CC 4C086
  • A61K31/422
  • .....not condensed and containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/423
  • .....condensed with carbocyclic rings [7] HB CC 4C086
  • A61K31/424
  • .....condensed with heterocyclic ring systems, e.g. clavulanic acid [7] HB CC 4C086
  • A61K31/4245
  • ....Oxadiazoles [7] HB CC 4C086
  • A61K31/425
  • ....Thiazoles [2,7] HB CC 4C086
  • A61K31/426
  • .....1,3-Thiazoles [7] HB CC 4C086
  • A61K31/427
  • .....not condensed and containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/428
  • .....condensed with carbocyclic rings [7] HB CC 4C086
  • A61K31/429
  • .....condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/43
  • ......Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula [figure], e.g. penicillins, penems [2,6] HB CC 4C086
  • A61K31/431
  • .......containing further heterocyclic ring systems, e.g. ticarcillin, azlocillin, oxacillin [7] HB CC 4C086
  • A61K31/433
  • ....Thiadiazoles [7] HB CC 4C086
  • A61K31/435
  • ...having six-membered rings with one nitrogen as the only ring hetero atom [2] HB CC 4C086
  • A61K31/4353
  • ....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/4355
  • .....the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom [7] HB CC 4C086
  • A61K31/436
  • .....the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin [7] HB CC 4C086
  • A61K31/4365
  • .....the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine [7] HB CC 4C086
  • A61K31/437
  • .....the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline [7] HB CC 4C086
  • A61K31/4375
  • .....the heterocyclic ring system containing a six-membered ring having nitrogen as a ring hetero atom, e.g. quinolizines, naphthyridines, berberine, vincamine [7] HB CC 4C086
  • A61K31/438
  • ....the ring being spiro-condensed with carbocyclic or heterocyclic ring systems [7] HB CC 4C086
  • A61K31/439
  • ....the ring forming part of a bridged ring system, e.g. quinuclidine (8-azabicyclo [3.2.1] octanes A61K 31/46) [7] HB CC 4C086
  • A61K31/44
  • ....Non-condensed pyridines; Hydrogenated derivatives thereof [2,7] HB CC 4C086
  • A61K31/4402
  • .....only substituted in position 2, e.g. pheniramine, bisacodyl [7] HB CC 4C086
  • A61K31/4406
  • .....only substituted in position 3, e.g. zimeldine (nicotinic acid A61K 31/455) [7] HB CC 4C086
  • A61K31/4409
  • .....only substituted in position 4, e.g. isoniazid, iproniazid [7] HB CC 4C086
  • A61K31/4412
  • .....having oxo groups directly attached to the heterocyclic ring [7] HB CC 4C086
  • A61K31/4415
  • .....Pyridoxine, i.e.vitamin B6 (pyridoxal phosphate A61K 31/675) [7] HB CC 4C086
  • A61K31/4418
  • .....having a carbocyclic ring directly attached to the heterocyclic ring, e.g. cyproheptadine [7] HB CC 4C086
  • A61K31/4422
  • .....1,4-Dihydropyridines, e.g. nifedipine, nicardipine [7] HB CC 4C086
  • A61K31/4425
  • .....Pyridinium derivatives, e.g. pralidoxime, pyridostigmine [7] HB CC 4C086
  • A61K31/4427
  • .....containing further heterocyclic ring systems [7] HB CC 4C086
  • A61K31/443
  • ......containing a five-membered ring with oxygen as a ring hetero atom [7] HB CC 4C086
  • A61K31/4433
  • ......containing a six-membered ring with oxygen as a ring hetero atom [7] HB CC 4C086
  • A61K31/4436
  • ......containing a heterocyclic ring having sulfur as a ring hetero atom [7] HB CC 4C086
  • A61K31/4439
  • ......containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole (nicotine A61K 31/465) [7] HB CC 4C086
  • A61K31/444
  • ......containing a six-membered ring with nitrogen as a ring hetero atom, e.g. amrinone [7] HB CC 4C086
  • A61K31/445
  • .....Non-condensed piperidines, e.g. piperocaine [2,7] HB CC 4C086
  • A61K31/4453
  • ......only substituted in position 1, e.g. propipocaine, diperodon [7] HB CC 4C086
  • A61K31/4458
  • ......only substituted in position 2, e.g. methylphenidate [7] HB CC 4C086
  • A61K31/4462
  • ......only substituted in position 3 [7] HB CC 4C086
  • A61K31/4465
  • ......only substituted in position 4 [7] HB CC 4C086
  • A61K31/4468
  • ......having a nitrogen atom directly attached in position 4, e.g. clebopride, fentanyl [7] HB CC 4C086
  • A61K31/45
  • ......having oxo groups directly attached to the heterocyclic ring, e.g. cycloheximide [2,7] HB CC 4C086
  • A61K31/451
  • ......having a carbocyclic ring directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine [7] HB CC 4C086
  • A61K31/4515
  • ......having a butyrophenone group in position 1, e.g. haloperidol (pipamperone A61K 31/4545) [7] HB CC 4C086
  • A61K31/452
  • ......Piperidinium derivatives (pancuronium A61K 31/58) [7] HB CC 4C086
  • A61K31/4523
  • ......containing further heterocyclic ring systems [7] HB CC 4C086
  • A61K31/4525
  • .......containing a five-membered ring with oxygen as a ring hetero atom [7] HB CC 4C086
  • A61K31/453
  • .......containing a six-membered ring with oxygen as a ring hetero atom [7] HB CC 4C086
  • A61K31/4535
  • .......containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen [7] HB CC 4C086
  • A61K31/454
  • .......containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone [7] HB CC 4C086
  • A61K31/4545
  • .......containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine [7] HB CC 4C086
  • A61K31/455
  • .....Nicotinic acid, i.e. niacin; Derivatives thereof, e.g. esters, amides [2] HB CC 4C086
  • A61K31/46
  • ....8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine [2] HB CC 4C086
  • A61K31/465
  • ....Nicotine; Derivatives thereof [2] HB CC 4C086
  • A61K31/47
  • ....Quinolines; Isoquinolines [2] HB CC 4C086
  • A61K31/4704
  • .....2-Quinolinones, e.g. carbostyril [7] HB CC 4C086
  • A61K31/4706
  • .....4-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine [7] HB CC 4C086
  • A61K31/4709
  • .....Non-condensed quinolines containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/472
  • .....Non-condensed isoquinolines, e.g. papaverine [7] HB CC 4C086
  • A61K31/4725
  • ......containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/473
  • .....ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines [7] HB CC 4C086
  • A61K31/4738
  • .....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/4741
  • ......condensed with ring systems having oxygen as a ring hetero atom, e.g. tubocuraran derivatives, noscapine, bicuculline [7] HB CC 4C086
  • A61K31/4743
  • ......condensed with ring systems having sulfur as a ring hetero atom [7] HB CC 4C086
  • A61K31/4745
  • ......condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenanthrolines (yohimbine derivatives, vinblastine A61K 31/475; ergoline derivatives A61K 31/48) [7] HB CC 4C086
  • A61K31/4747
  • .....spiro-condensed [7] HB CC 4C086
  • A61K31/4748
  • .....forming part of bridged ring systems (strychnine A61K 31/475; morphinan derivatives A61K 31/485) [7] HB CC 4C086
  • A61K31/475
  • .....having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine (vincamine A61K 31/4375) [2,7] HB CC 4C086
  • A61K31/48
  • .....Ergoline derivatives, e.g. lysergic acid, ergotamine [2,7] HB CC 4C086
  • A61K31/485
  • .....Morphinan derivatives, e.g. morphine, codeine [2,7] HB CC 4C086
  • A61K31/49
  • .....Cinchonan derivatives, e.g. quinine [2,7] HB CC 4C086
  • A61K31/495
  • ...having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine (A61K 31/48 takes precedence) [2] HB CC 4C086
  • A61K31/496
  • ....Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin [2006.01] HB CC 4C086
  • A61K31/4965
  • ....Non-condensed pyrazines [7] HB CC 4C086
  • A61K31/497
  • .....containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/498
  • ....Pyrazines or piperazines ortho- or peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine [7] HB CC 4C086
  • A61K31/4985
  • ....Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/499
  • ....Spiro-condensed pyrazines or piperazines [7] HB CC 4C086
  • A61K31/4995
  • ....Pyrazines or piperazines forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/50
  • ....Pyridazines; Hydrogenated pyridazines [2,7] HB CC 4C086
  • A61K31/501
  • .....not condensed and containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/502
  • .....ortho- or peri-condensed with carbocyclic ring systems, e.g. cinnoline, phthalazine [7] HB CC 4C086
  • A61K31/5025
  • .....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/503
  • .....spiro-condensed [7] HB CC 4C086
  • A61K31/504
  • .....forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/505
  • ....Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim [2,7] HB CC 4C086
  • A61K31/506
  • .....not condensed and containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/51
  • ......Thiamines, e.g. vitamin B1 [2] HB CC 4C086
  • A61K31/513
  • .....having oxo groups directly attached to the heterocyclic ring, e.g. cytosine [7] HB CC 4C086
  • A61K31/515
  • ......Barbituric acids; Derivatives thereof, e.g. sodium pentobarbital [2] HB CC 4C086
  • A61K31/517
  • .....ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine [7] HB CC 4C086
  • A61K31/519
  • .....ortho- or peri-condensed with heterocyclic rings [7] HB CC 4C086
  • A61K31/52
  • ......Purines, e.g. adenine [2,7] HB CC 4C086
  • A61K31/522
  • .......having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir [7, 2006.01] HB CC 4C086
  • A61K31/525
  • ......Isoalloxazines, e.g. riboflavins, vitamin B2 [2] HB CC 4C086
  • A61K31/527
  • .....spiro-condensed [7] HB CC 4C086
  • A61K31/529
  • .....forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/53
  • ...having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine (melarsoprol A61K 31/555) [2] HB CC 4C086
  • A61K31/535
  • ...having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines [2] HB CC 4C086
  • A61K31/5355
  • ....Non-condensed oxazines containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/536
  • ....ortho- or peri-condensed with carbocyclic ring systems [7] HB CC 4C086
  • A61K31/5365
  • ....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/537
  • ....spiro-condensed or forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/5375
  • ....1,4-Oxazines, e.g. morpholine [7] HB CC 4C086
  • A61K31/5377
  • .....not condensed and containing further heterocyclic rings, e.g. timolol [7] HB CC 4C086
  • A61K31/538
  • .....ortho- or peri-condensed with carbocyclic ring systems [7] HB CC 4C086
  • A61K31/5383
  • .....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/5386
  • .....spiro-condensed or forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/539
  • ....having two or more oxygen atoms in the same ring, e.g dioxazines [7] HB CC 4C086
  • A61K31/5395
  • ....having two or more nitrogen atoms in the same ring, e.g. oxadiazines [7] HB CC 4C086
  • A61K31/54
  • ...having six-membered rings with at least one nitrogen and at least one sulfur as the ring hetero atoms, e.g. sulthiame [2] HB CC 4C086
  • A61K31/541
  • ....Non-condensed thiazines containing further heterocyclic rings [7] HB CC 4C086
  • A61K31/5415
  • ....ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam [7] HB CC 4C086
  • A61K31/542
  • ....ortho- or peri-condensed with heterocyclic ring systems [7] HB CC 4C086
  • A61K31/545
  • .....Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula [figure], e.g. cephalosporins, cefaclor, cephalexine [2,6] HB CC 4C086
  • A61K31/546
  • ......containing further heterocyclic rings, e.g. cephalothin [7] HB CC 4C086
  • A61K31/547
  • ....spiro-condensed or forming part of bridged ring systems [7] HB CC 4C086
  • A61K31/548
  • ....having two or more sulfur atoms in the same ring [7] HB CC 4C086
  • A61K31/549
  • ....having two or more nitrogen atoms in the same ring, e.g. hydrochlorothiazide [7] HB CC 4C086
  • A61K31/55
  • ...having seven-membered rings, e.g. azelastine, pentylenetetrazole [2] HB CC 4C086
  • A61K31/551
  • ....having two nitrogens as ring hetero atoms, e.g. clozapine, dilazep [7] HB CC 4C086
  • A61K31/5513
  • .....1,4-Benzodiazepines, e.g. diazepam [7] HB CC 4C086
  • A61K31/5517
  • ......condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam [7] HB CC 4C086
  • A61K31/553
  • ....having at least one nitrogen and at least one oxygen as ring hetero atoms, e.g. loxapine, staurosporine [7] HB CC 4C086
  • A61K31/554
  • ....having at least one nitrogen and at least one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem [7] HB CC 4C086
  • A61K31/555
  • ..containing heavy metals, e.g. hemin, hematin, melarsoprol [2] HB CC 4C086
  • A61K31/557
  • .Eicosanoids, e.g. leukotrienes [3,7] HB CC 4C086
  • A61K31/5575
  • ..having a cyclopentane ring, e.g. prostaglandin E2, prostaglandin F2-alpha [7] HB CC 4C086
  • A61K31/5578
  • ..having a pentalene ring system, e.g. carbacyclin, iloprost [7] HB CC 4C086
  • A61K31/558
  • ..having heterocyclic rings containing oxygen as the only ring hetero atom, e.g. thromboxanes [7] HB CC 4C086
  • A61K31/5585
  • ...having five-membered rings containing oxygen as the only ring hetero atom, e.g. prostacyclin [7] HB CC 4C086
  • A61K31/559
  • ..having heterocyclic rings containing hetero atoms other than oxygen [7] HB CC 4C086
  • A61K31/56
  • .Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids HB CC 4C086
  • A61K31/565
  • ..not substituted in position 17 beta by a carbon atom, e.g. oestrane, oestradiol [2] HB CC 4C086
  • A61K31/566
  • ...having an oxo group in position 17, e.g. oestrone [7] HB CC 4C086
  • A61K31/567
  • ...substituted in position 17 alpha, e.g. mestranol, norethandrolone [7] HB CC 4C086
  • A61K31/568
  • ...substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstane, testosterone [7] HB CC 4C086
  • A61K31/5685
  • ....having an oxo group in position 17, e.g. androsterone [7] HB CC 4C086
  • A61K31/569
  • ....substituted in position 17 alpha, e.g. ethisterone [7] HB CC 4C086
  • A61K31/57
  • ..substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone [2006.01] HB CC 4C086
  • A61K31/573
  • ...substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone [2006.01] HB CC 4C086
  • A61K31/575
  • ..substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol [2] HB CC 4C086
  • A61K31/58
  • ..containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin (digitoxin A61K 31/704) [2006.01] HB CC 4C086
  • A61K31/585
  • ...containing lactone rings, e.g. oxandrolone, bufalin [2] HB CC 4C086
  • A61K31/59
  • .Compounds containing 9,10-seco-cyclopenta[a]hydro- phenanthrene ring systems [2] HB CC 4C086
  • A61K31/592
  • ..9,10-Secoergostane derivatives, e.g. ergocalciferol, vitamin D2 [7] HB CC 4C086
  • A61K31/593
  • ..9,10-Secocholestane derivatives, e.g. cholecalciferol, vitamin D3 [7] HB CC 4C086
  • A61K31/60
  • .Salicylic acid; Derivatives thereof [2] HB CC 4C086
  • A61K31/603
  • ..having further aromatic rings, e.g. diflunisal [7] HB CC 4C086
  • A61K31/606
  • ..having amino groups [7] HB CC 4C086
  • A61K31/609
  • ..Amides, e.g. salicylamide [7] HB CC 4C086
  • A61K31/612
  • ..having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid (fosfosal A61K 31/661) [7] HB CC 4C086
  • A61K31/616
  • ...by carboxylic acids, e.g. acetylsalicylic acid [7] HB CC 4C086
  • A61K31/618
  • ..having the carboxyl group in position 1 esterified, e.g. salsalate [7] HB CC 4C086
  • A61K31/621
  • ...having the hydroxy group in position 2 esterified, e.g. benorylate [7] HB CC 4C086
  • A61K31/625
  • ..having heterocyclic substituents, e.g. 4-salicyloylmorpholine (sulfasalazine A61K 31/635) [2,7] HB CC 4C086
  • A61K31/63
  • .Compounds containing para-N-benzene- sulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonohydrazide [2] HB CC 4C086
  • A61K31/635
  • ..having a heterocyclic ring, e.g. sulfadiazine [2] HB CC 4C086
  • A61K31/64
  • .Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide [2] HB CC 4C086
  • A61K31/65
  • .Tetracyclines [2] HB CC 4C086
  • A61K31/655
  • .Azo (—N=N—), diazo (=N2), azoxy (3) or diazoamino (—N=N—N<) compounds [2] HB CC 4C086
  • A61K31/66
  • .Phosphorus compounds [2] HB CC 4C086
  • A61K31/661
  • ..Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion [7] HB CC 4C086
  • A61K31/6615
  • ...Compounds having two or more esterified phosphorus acid groups, e.g. inositol triphosphate, phytic acid [7] HB CC 4C086
  • A61K31/662
  • ..Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon [7] HB CC 4C086
  • A61K31/663
  • ...Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid [7] HB CC 4C086
  • A61K31/664
  • ..Amides of phosphorus acids [7] HB CC 4C086
  • A61K31/665
  • ..having oxygen as a ring hetero atom, e.g. fosfomycin [2] HB CC 4C086
  • A61K31/67
  • ..having sulfur as a ring hetero atom [2] HB CC 4C086
  • A61K31/675
  • ..having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate [2] HB CC 4C086
  • A61K31/683
  • ..Diesters of a phosphorus acid with two hydroxy compounds, e.g. phosphatidylinositols [7] HB CC 4C086
  • A61K31/685
  • ...one of the hydroxy compounds having nitrogen atoms, e.g. phosphatidylserine, lecithin [2,7] HB CC 4C086
  • A61K31/688
  • ...both hydroxy compounds having nitrogen atoms, e.g. sphingomyelins [7] HB CC 4C086
  • A61K31/69
  • .Boron compounds [2] HB CC 4C086
  • A61K31/695
  • .Silicon compounds [2] HB CC 4C086
  • A61K31/70
  • .Carbohydrates; Sugars; Derivatives thereof (sorbitol A61K 31/047) HB CC 4C086
  • A61K31/7004
  • ..Monosaccharides having only carbon, hydrogen and oxygen atoms [7] HB CC 4C086
  • A61K31/7008
  • ..Compounds having an amino group directly attached to a carbon atom of the saccharide radical, e.g. D-galactosamine, ranimustine [7] HB CC 4C086
  • A61K31/7012
  • ..Compounds having a free or esterified carboxyl group attached, directly or through a carbon chain, to a carbon atom of the saccharide radical, e.g. glucuronic acid, neuraminic acid (gluconic acid A61K 31/191; ascorbic acid A61K 31/375) [7] HB CC 4C086
  • A61K31/7016
  • ..Disaccharides, e.g. lactose, lactulose (lactobionic acid A61K 31/7032) [7] HB CC 4C086
  • A61K31/702
  • ..Oligosaccharides, i.e. having three to five saccharide radicals attached to each other by glycosidic linkages [7] HB CC 4C086
  • A61K31/7024
  • ..Esters of saccharides [7] HB CC 4C086
  • A61K31/7028
  • ..Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages [7] HB CC 4C086
  • A61K31/7032
  • ...attached to a polyol, i.e. compounds having two or more free or esterified hydroxy groups, including the hydroxy group involved in the glycosidic linkage, e.g. monoglucosyl-diacylglycerides, lactobionic acid, gangliosides [7] HB CC 4C086
  • A61K31/7034
  • ...attached to a carbocyclic compound, e.g. phloridzin [7] HB CC 4C086
  • A61K31/7036
  • ....having at least one amino group directly attached to the carbocyclic ring, e.g. streptomycin, gentamycin, amikacin, validamycin, fortimicins [7] HB CC 4C086
  • A61K31/704
  • ....attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin, digitoxin [7] HB CC 4C086
  • A61K31/7042
  • ..Compounds having saccharide radicals and heterocyclic rings [7] HB CC 4C086
  • A61K31/7048
  • ...having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin [7] HB CC 4C086
  • A61K31/7052
  • ...having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides [7] HB CC 4C086
  • A61K31/7056
  • ....containing five-membered rings with nitrogen as a ring hetero atom [7] HB CC 4C086
  • A61K31/706
  • ....containing six-membered rings with nitrogen as a ring hetero atom [7] HB CC 4C086
  • A61K31/7064
  • .....containing condensed or non-condensed pyrimidines [7] HB CC 4C086
  • A61K31/7068
  • ......having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid [7] HB CC 4C086
  • A61K31/7072
  • .......having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine [7] HB CC 4C086
  • A61K31/7076
  • ......containing purines, e.g. adenosine, adenylic acid [7] HB CC 4C086
  • A61K31/708
  • .......having oxo groups directly attached to the purine ring system, e.g. guanosine, guanylic acid [7] HB CC 4C086
  • A61K31/7084
  • ..Compounds having two nucleosides or nucleotides, e.g. nicotinamide-adenine dinucleotide, flavine-adenine dinucleotide [7] HB CC 4C086
  • A61K31/7088
  • ..Compounds having three or more nucleosides or nucleotides [7] HB CC 4C086
  • A61K31/7105
  • ...Natural ribonucleic acids, i.e. containing only riboses attached to adenine, guanine, cytosine or uracil and having 3'-5' phosphodiester links [7] HB CC 4C086
  • A61K31/711
  • ...Natural deoxyribonucleic acids, i.e. containing only 2'-deoxyriboses attached to adenine, guanine, cytosine or thymine and having 3'-5' phosphodiester links [7] HB CC 4C086
  • A61K31/7115
  • ...Nucleic acids or oligonucleotides having modified bases, i.e. other than adenine, guanine, cytosine, uracil or thymine [7] HB CC 4C086
  • A61K31/712
  • ...Nucleic acids or oligonucleotides having modified sugars, i.e. other than ribose or 2'-deoxyribose [7] HB CC 4C086
  • A61K31/7125
  • ...Nucleic acids or oligonucleotides having modified internucleoside linkage, i.e. other than 3'-5' phosphodiesters [7] HB CC 4C086
  • A61K31/713
  • ...Double-stranded nucleic acids or oligonucleotides [7] HB CC 4C086
  • A61K31/7135
  • ..Compounds containing heavy metals [7] HB CC 4C086
  • A61K31/714
  • ...Cobalamins, e.g. cyanocobalamin, vitamin B12 [7] HB CC 4C086
  • A61K31/715
  • ..Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters [2] HB CC 4C086
  • A61K31/716
  • ...Glucans [7] HB CC 4C086
  • A61K31/717
  • ....Celluloses [7] HB CC 4C086
  • A61K31/718
  • ....Starch or degraded starch, e.g. amylose, amylopectin [7] HB CC 4C086
  • A61K31/719
  • ....Pullulans [7] HB CC 4C086
  • A61K31/721
  • ....Dextrans [7] HB CC 4C086
  • A61K31/722
  • ....Chitin; Chitosan [7] HB CC 4C086
  • A61K31/723
  • ....Xanthans [7] HB CC 4C086
  • A61K31/724
  • ....Cyclodextrins [7] HB CC 4C086
  • A61K31/726
  • ...Glycosaminoglycans, i.e. mucopolysaccharides (chondroitin sulfate, dermatan sulfate A61K 31/737) [7] HB CC 4C086
  • A61K31/727
  • ....Heparin; Heparan [7] HB CC 4C086
  • A61K31/728
  • ....Hyaluronic acid [7] HB CC 4C086
  • A61K31/729
  • ...Agar; Agarose; Agaropectin [7] HB CC 4C086
  • A61K31/731
  • ...Carrageenans [7] HB CC 4C086
  • A61K31/732
  • ...Pectin [7] HB CC 4C086
  • A61K31/733
  • ...Fructosans, e.g. inulin [7] HB CC 4C086
  • A61K31/734
  • ...Alginic acid [7] HB CC 4C086
  • A61K31/736
  • ...Glucomannans or galactomannans, e.g locust bean gum, guar gum [7] HB CC 4C086
  • A61K31/737
  • ...Sulfated polysaccharides, e.g. chondroitin sulfate, dermatan sulfate (A61K 31/727 takes precedence) [7] HB CC 4C086
  • A61K31/738
  • ...Cross-linked polysaccharides [7] HB CC 4C086
  • A61K31/739
  • ...Lipopolysaccharides [7] HB CC 4C086
  • A61K31/74
  • .Synthetic polymeric materials [2] HB CC 4C086
  • A61K31/745
  • ..Polymers of hydrocarbons [2] HB CC 4C086
  • A61K31/75
  • ...of ethene [2] HB CC 4C086
  • A61K31/755
  • ..Polymers containing halogen [2] HB CC 4C086
  • A61K31/76
  • ...of vinyl chloride [2] HB CC 4C086
  • A61K31/765
  • ..Polymers containing oxygen [2] HB CC 4C086
  • A61K31/77
  • ...of oxiranes [2] HB CC 4C086
  • A61K31/775
  • ...Phenolic resins [2] HB CC 4C086
  • A61K31/78
  • ...of acrylic acid or derivatives thereof [2] HB CC 4C086
  • A61K31/785
  • ..Polymers containing nitrogen [2] HB CC 4C086
  • A61K31/787
  • ...containing heterocyclic rings having nitrogen as a ring hetero atom [7] HB CC 4C086
  • A61K31/79
  • ....Polymers of vinyl pyrrolidone [2] HB CC 4C086
  • A61K31/795
  • ..Polymers containing sulfur [2] HB CC 4C086
  • A61K31/80
  • ..Polymers containing hetero atoms not provided for in groups A61K 31/755-A61K 31/795 [2] HB CC 4C086
    TOP